Regioselective alkylation of 1,3,4,5-tetrahydrobenzo[d]azepin-2-one and biological evaluation of the resulting alkylated products as potentially selective $$\hbox {5-HT}_{\mathrm{2C}}$$ 5-HT 2 C agonists-Reference-Cited by-同舟云学术

Regioselective alkylation of 1,3,4,5-tetrahydrobenzo[d]azepin-2-one and biological evaluation of the resulting alkylated products as potentially selective $$\hbox {5-HT}_{\mathrm{2C}}$$ 5-HT 2 C agonists

Published:2015-04-28 Issue:4 Volume:19 Page:653-667
ISSN:1381-1991
Container-title:Molecular Diversity
language:en
Short-container-title:Mol Divers

Author:

Prajapati Navnit,Giridhar Rajani,Sinha Anshuman,Kanhed Ashish M.,Yadav Mange Ram

Publisher

Springer Science and Business Media LLC

Subject

Inorganic Chemistry,Organic Chemistry,Physical and Theoretical Chemistry,Drug Discovery,Molecular Biology,General Medicine,Information Systems,Catalysis

Link

http://link.springer.com/content/pdf/10.1007/s11030-015-9600-8.pdf

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4. Bello NT, Liang NC (2011) The use of serotonergic drugs to treat obesity—is there any hope? Drug Des Devel Ther 5:95–109. doi: 10.2147/DDDT.S11859

5. Sheridan MH (2013) Lorcaserin: a review of its use in chronic weight management. Drugs 73:463–473. doi: 10.1007/s40265-013-0035-1

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2. 3-Substituted 1-methyl-3-benzazepin-2-ones as 5-HT2C receptor agonists;RSC Advances;2015