The histamine H1-receptor antagonist binding site. Part I: Active conformation of cyproheptadine-Reference-Cited by-同舟云学术

The histamine H1-receptor antagonist binding site. Part I: Active conformation of cyproheptadine

Published:1991-08 Issue:4 Volume:5 Page:357-370
ISSN:0920-654X
Container-title:Journal of Computer-Aided Molecular Design
language:en
Short-container-title:J Computer-Aided Mol Des

Author:

van Drooge Marc J.,Donné-op den Kelder Gabriëlle M.,Timmerman Hendrik

Publisher

Springer Science and Business Media LLC

Subject

Physical and Theoretical Chemistry,Computer Science Applications,Drug Discovery

Link

http://link.springer.com/content/pdf/10.1007/BF00126668.pdf

Reference25 articles.

1. Nauta, W.Th. and Rekker, R.F., In Roche e, Silva (Ed.) Handbook of Experimental Pharmacology, Part 18/2 Springer, Berlin, 1978, pp. 215?249.

2. Waringa, C.G., Rekker, R.F. and Nauta, W.Th., Eur. J. Med. Chem., 10 (1975) 349.

3. Harms, A.F., Hespe, W., Nauta, W.Th., Rekker, R.F., Timmerman, H. and De, Vries, J., In Ariëns, E.J. (Ed.), Drug Design, Vol. VI, Academic Press, New York, 1975, pp. 1?80.

4. Durant, G.J., Ganellin, C.R., Griffiths, R., Harvey, C.A., Owen, D.A.A. and Sach, G.S., Adv. Biosci., 51 (1985) 3.

5. Iemura, R. and Ohtaka, H., Chem. Pharm. Bull., 37 (1989), 967.

Cited by 9 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Prescribed drugs containing nitrogen heterocycles: an overview;RSC Advances;2020

2. Synthesis and antihistamine evaluations of novel loratadine analogues;Bioorganic & Medicinal Chemistry Letters;2011-08

3. Comparative structure–activity relationships of benztropine analogues at the dopamine transporter and histamine H1 receptors;Bioorganic & Medicinal Chemistry;2006-06

4. Delineation of Receptor-Ligand Interactions at the Human Histamine H1 Receptor by a Combined Approach of Site-Directed Mutagenesis and Computational Techniques - or - How to Bind the H1 Receptor;Archiv der Pharmazie;2005-06

5. Computer-Assisted Comparison of the Structural and Electronic Dispositions of Ebastine and Terfenadine;Drug Safety;1999