Inhibiting a promiscuous GPCR: iterative discovery of bitter taste receptor ligands-Reference-Cited by-同舟云学术

Inhibiting a promiscuous GPCR: iterative discovery of bitter taste receptor ligands

Published:2023-04 Issue:4 Volume:80 Page:
ISSN:1420-682X
Container-title:Cellular and Molecular Life Sciences
language:en
Short-container-title:Cell. Mol. Life Sci.

Author:

Fierro Fabrizio^ORCID,Peri Lior,Hübner Harald,Tabor-Schkade Alina,Waterloo Lukas,Löber Stefan,Pfeiffer Tara,Weikert Dorothee,Dingjan Tamir,Margulis Eitan,Gmeiner Peter,Niv Masha Y^ORCID

Funder

Deutsche Forschungsgemeinschaft

Lady Davis Fellowship Trust, Hebrew University of Jerusalem

Center for Nanoscience and Nanotechnology, Hebrew University of Jerusalem

Israel Science Foundation

Publisher

Springer Science and Business Media LLC

Subject

Cell Biology,Cellular and Molecular Neuroscience,Pharmacology,Molecular Biology,Molecular Medicine

Link

https://link.springer.com/content/pdf/10.1007/s00018-023-04765-0.pdf

Reference67 articles.

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3. Chan WK, Zhang H, Yang J, Brender JR et al (2015) GLASS: a comprehensive database for experimentally validated GPCR-ligand associations. Bioinformatics 31(18):3035–3042

4. Sriram K, Insel PA (2018) G protein-coupled receptors as targets for approved drugs: how many targets and how many drugs? Mol Pharmacol 93(4):251–258

5. Dagan-Wiener A, Di Pizio A, Nissim I, Bahia MS et al (2019) BitterDB: taste ligands and receptors database in 2019. Nucleic Acids Res 47(D1):D1179–D1185

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