Relation between pharmacological response and receptor binding with histamine blocking drugs. Irreversible antagonism of three analogues of mifentidine on right atrium and cerebral cortex of the guinea-pig-Reference-Cited by-同舟云学术

Relation between pharmacological response and receptor binding with histamine blocking drugs. Irreversible antagonism of three analogues of mifentidine on right atrium and cerebral cortex of the guinea-pig

Published:1987-06 Issue:1-2 Volume:21 Page:41-48
ISSN:0065-4299
Container-title:Agents and Actions
language:en
Short-container-title:Agents and Actions

Author:

Kramer K.,Bast A.,Timmerman H.

Publisher

Springer Science and Business Media LLC

Subject

Pharmacology (medical),Toxicology,Pharmacology,Immunology

Link

http://link.springer.com/content/pdf/10.1007/BF01974919.pdf

Reference19 articles.

1. A. S. F. Ash and H. O. Schild,Receptors mediating some actions of histamine. Br. J. Pharmac. Chemother.27, 427–439 (1966).

2. J. W. Black, W. A. M. Duncan, C. J. Durant, C. R. Ganellin and M. E. Parsons,Definition and antagonism of histamine, H 2 -receptor. Nature236, 385–390 (1972).

3. M. W. McCulloch, I. C. Medgett, M. J. Rand and D. F. Story,Structure-activity relationship of imidazoline derivatives related to clonidine at histamine H 2 -receptors in guinea-pig isolated atria. Br. J. Pharmac.69, 397–405 (1980).

4. K. Ozawa, Y. Nomura and T. Segawa,Mechanism of Cu 2+ -induced elevation of [3 H]-cimetidine binding to membranes in rat brain. Neurochem. Int.7, 435–440 (1985).

5. W. P. Burhard,Histamine H 2 -receptor binding with [3 H]-cimetidine in brain. Eur. J. Pharmac.50, 449–450 (1978).

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