Phenotypic assessment and ligand screening of ETA/ETB receptors with label-free dynamic mass redistribution assay

Author:

Qu Lala,Zhang XiuliORCID,Wang Jixia,Zhou Han,Hou Tao,Wei Lai,Xu Fangfang,Liang Xinmiao

Funder

The State Key Program of National Natural Science of China

Project of National Science Foundation of China

The innovation program of science and research from DICP, CAS

Innovation platform for the development and construction of special project of Key Laboratory of Tibetan Medicine Research of Qinghai Province

Publisher

Springer Science and Business Media LLC

Subject

Pharmacology,General Medicine

Reference48 articles.

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2. Christensen HB, Gloriam DE, Pedersen DS, Cowland JB, Borregaard N, Brauner-Osborne H (2017) Applying label-free dynamic mass redistribution assay for studying endogenous FPR1 receptor signalling in human neutrophils. J Pharmacol Toxicol Methods 88(Pt 1):72–78. https://doi.org/10.1016/j.vascn.2017.07.003

3. Clozel M, Breu V, Gray GA, Kalina B, Loffler BM, Burri K, Cassal JM, Hirth G, Muller M, Neidhart W, Ramuz H (1994) Pharmacological characterization of Bosentan, a new potent orally-active nonpeptide endothelin receptor antagonist. J Pharmacol Exp Ther 270(1):228–235

4. Davenport AP, Hyndman KA, Dhaun N, Southan C, Kohan DE, Pollock JS, Pollock DM, Webb DJ, Maguire JJ (2016) Endothelin. Pharmacol Rev 68(2):357–418. https://doi.org/10.1124/pr.115.011833

5. Deng H, Fang Y (2013) The three catecholics benserazide, catechol and pyrogallol are GPR35 agonists. Pharmaceuticals (Basel, Switzerland) 6(4):500–509. https://doi.org/10.3390/ph6040500

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