Characterization of a novel, brain-penetrating CB1 receptor inverse agonist: metabolic profile in diet-induced obese models and aspects of central activity-Reference-Cited by-同舟云学术

Characterization of a novel, brain-penetrating CB1 receptor inverse agonist: metabolic profile in diet-induced obese models and aspects of central activity

Published:2011-09-25 Issue:6 Volume:384 Page:565-581
ISSN:0028-1298
Container-title:Naunyn-Schmiedeberg's Archives of Pharmacology
language:en
Short-container-title:Naunyn-Schmiedeberg's Arch Pharmacol

Author:

Jacobson Laura H.,Commerford S. Renee,Gerber Sarah P.,Chen Yu Alice,Dardik Beatriz,Chaperon Frederique,Schwartzkopf Chad,Nguyen-Tran Van,Hollenbeck Thomas,McNamara Peter,He Xiaohui,Liu Hong,Seidel H. Martin,Jaton Anne-Liese,Gromada Jesper,Teixeira Sandra

Publisher

Springer Science and Business Media LLC

Subject

Pharmacology,General Medicine

Link

http://link.springer.com/content/pdf/10.1007/s00210-011-0686-y.pdf

Reference47 articles.

1. Aronne LJ, Tonstad S, Moreno M, Gantz I, Erondu N, Suryawanshi S, Molony C, Sieberts S, Nayee J, Meehan AG, Shapiro D, Heymsfield SB, Kaufman KD, Amatruda JM (2010) A clinical trial assessing the safety and efficacy of taranabant, a CB1R inverse agonist, in obese and overweight patients: a high-dose study. Int J Obes (Lond) 34(5):919–935

2. Banker MJ, Clark TH, Williams JA (2003) Development and validation of a 96-well equilibrium dialysis apparatus for measuring plasma protein binding. J Pharm Sci 92:967–974

3. Bellocchio L, Lafenêtre P, Cannich A, Cota D, Puente N, Grandes P, Chaouloff F, Piazza PV, Marsicano G (2010) Bimodal control of stimulated food intake by the endocannabinoid system. Nat Neurosci 13(3):281–283

4. Cannich A, Wotjak CT, Kamprath K, Hermann H, Lutz B, Marsicano G (2004) CB1 cannabinoid receptors modulate kinase and phosphatase activity during extinction of conditioned fear in mice. Learn Mem 11:625–632

5. Chaperon F, Thiébot MH (1999) Behavioral effects of cannabinoid agents in animals. Crit Rev Neurobiol 13:243–281

Cited by 6 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Effects of Cannabinoid Agonists and Antagonists on Sleep in Laboratory Animals;Advances in Experimental Medicine and Biology;2021

2. Sex differences in mouse models of fear inhibition: Fear extinction, safety learning, and fear–safety discrimination;British Journal of Pharmacology;2019-04-15

3. Endocannabinoid Signaling Regulates Sleep Stability;PLOS ONE;2016-03-31

4. Modulation of food consumption and sleep–wake cycle in mice by the neutral CB1 antagonist ABD459;Behavioural Pharmacology;2015-04

5. Interrelationship of CB1R and OBR pathways in regulation of metabolic, neuroendocrine, and behavioral responses to food restriction and voluntary wheel running;Journal of Applied Physiology;2014-07-15