Prodrug enzymes and their applications in image-guided therapy of cancer: tracking prodrug enzymes to minimize collateral damage

Author:

Penet Marie-France,Chen Zhihang,Li Cong,Winnard Paul T.,Bhujwalla Zaver M.

Publisher

Springer Science and Business Media LLC

Subject

Pharmaceutical Science

Reference36 articles.

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2. Mahato R, et al. Prodrugs for improving tumor targetability and efficiency. Adv Drug Deliv Rev. 2011;63(8):659–70. PMCID: 3132824.

3. Sharma SK, et al. Sustained tumor regression of human colorectal cancer xenografts using a multifunctional mannosylated fusion protein in antibody-directed enzyme prodrug therapy. Clin Cancer Res. 2005;11(2 Pt 1):814–25.

4. Bhatia J, et al. Catalytic activity of an in vivo tumor targeted anti-CEA scFv::carboxypeptidase G2 fusion protein. Int J Cancer. 2000;85(4):571–7.

5. Longley DB, et al. 5-Fluorouracil: mechanisms of action and clinical strategies. Nat Rev Cancer. 2003;3(5):330–8.

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