Preparation and bioevaluation of [99mTcN]2+-labeled tetrameric complex of E-c(RGDfK)2 as a radiotracer for imaging αvβ3 integrins in tumors

Author:

Guleria Mohini,Ghosh Subhajit,Das Tapas,Sarma Haladhar Dev,Banerjee Sharmila

Funder

Bhabha Atomic Research Centre

Publisher

Springer Science and Business Media LLC

Subject

Health, Toxicology and Mutagenesis,Public Health, Environmental and Occupational Health,Spectroscopy,Pollution,Radiology Nuclear Medicine and imaging,Nuclear Energy and Engineering,Analytical Chemistry

Reference38 articles.

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2. Brooks PC, Clark RAF, Cheresh DA (1994) Requirement of vascular integrin αvβ3 for angiogenesis. Science 264:569–571

3. Gasparini G, Brooks PC, Biganzoli E, Bonoldi E, Dirix LY, Ranieri G, Miceli R, Cheresh DA (1998) Vascular integrin αvβ3 a new prognostic indicator in breast cancer. Clin Cancer Res 4:2625–2634

4. Albelda SM, Mette SA, Elder DE, Stewart RM, Damjanovich L, Herlyn M, Buck CA (1990) Integrin distribution in malignant melanoma: association of the β 3 subunit with tumor progression. Cancer Res 50:6757–6764

5. Sengupta S, Chattopadhyay N, Mitra A, Ray S, Dasgupta S, Chatterjee A (2001) Role of αvβ3 integrin receptors in breast tumor. J Exp Clin Cancer Res 20:585–590

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