The anxiolytic-like activity of GR159897, a non-peptide NK2 receptor antagonist, in rodent and primate models of anxiety
Author:
Publisher
Springer Science and Business Media LLC
Subject
Pharmacology
Link
http://link.springer.com/content/pdf/10.1007/BF02245629.pdf
Reference32 articles.
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3. Beresford IJM, Sheldrick RLG, Ball DI, Turpin MP, Walsh DM, Hawcock AB, Coleman RA, Hagan RM, Tyers MB (1995) GR159897, a potent non-peptide antagonist at tachykinin NK2 receptors. Eur J pharmacol 272:241–248
4. Bradwejn J, Koszycki D, Du Tertre AC, Van Megen H, Den Boer J, Westenberg H, Annable L (1994) The panicogenic effects of cholecystokinin-tetrapeptide are antagonized by L-365,260, a central cholecystokinin receptor antagonist, in patients with a panic disorder. Arch Gen Psychiatry 51:486–493
5. Cooper AWJ, Adams HS, Bell R, Gore PM, McElroy AB, Pritchard JM, Smith PW, Ward P (1994) GR159897 and related analogues as highly potent, orally active non-peptide neurokinin NK2 receptor antagonists. Bioorganic Med Chem Lett 4:1951–1956
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