Phase II trial of pyrazoloacridine (NSC#366140) in patients with metastatic breast cancer

Author:

Ramaswamy Bhuvaneswari,Mrozek Ewa,Kuebler John Philip,Bekaii-Saab Tanios,Kraut Eric H.

Publisher

Springer Science and Business Media LLC

Subject

Pharmacology (medical),Pharmacology,Oncology

Reference19 articles.

1. Adjei AA, Charron M, Rowinsky EK et al (1998) Effect of pyrazoloacridine (NSC 366140) on DNA topoisomerases I and II. Clin Cancer Res 4:683–691

2. Sebolt J, Havlick M, Hamelehle K et al (1989) Activity of the pyrazoloacridines against multidrug-resistant tumor cells. Cancer Chemother Pharmacol 24:219–224

3. Sebolt JS, Scavone SV, Pinter CD et al (1987) Pyrazoloacridines, a new class of anticancer agents with selectivity against solid tumors in vitro. Cancer Res 47:4299–4304

4. Grem JL, Politi PM, Berg SL et al (1996) Cytotoxicity and DNA damage associated with pyrazoloacridine in MCF-7 breast cancer cells. Biochem Pharmacol 51:1649–1659

5. Jackson RC, Sebolt JS, Shillis JL et al (1990) The pyrazoloacridines: approaches to the development of a carcinoma-selective cytotoxic agent. Cancer Invest 8:39–47

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