Saturable elimination and saturable protein binding account for flavone acetic acid pharmacokinetics

Author:

Relling Mary V.,Evans Robert R.,Groom Steven,Crom William R.,Pratt Charles B.

Publisher

Springer Science and Business Media LLC

Subject

Pharmacology (medical),General Pharmacology, Toxicology and Pharmaceutics

Reference21 articles.

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2. J. Cummings and J. F. Smyth. Flavone 8-acetic acid: Our current understanding of its mechanism of action in solid tumours.Cancer Chemother. and Pharmacol. 24:269–272 (1989).

3. C. B. Pratt, M. V. Relling, W. H. Meyer, E. C. Douglass, S. J. Kellie, and L. Avery. Phase I study of flavone acetic acid (NSC 347512, LM975) in patients with pediatric malignant solid tumors.Am. J. Clin. Oncol. 14:483–486 (1991).

4. R. B. Weiss, R. F. Green, R. D. Knight, J. M. Collins, J. J. Pelosi, A. Sulkes, and G. A. Curt. Phase I and clinical pharmacology study of intravenous flavone acetic acid (NSC 347512).Cancer Res. 48:5878–5882 (1988).

5. D. J. Kerr, S. B. Kaye, J. Cassidy, C. Bradley, E. M. Rankin, L. Adams, A. Setanoians, T. Young, G. Forrest, M. Soukop, and M. Clavel. Phase I and pharmacokinetic study of flavone acetic acid.Cancer Res. 47:6776–6781 (1987).

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