Properties Influencing the Relative Binding Affinity of Pteroate Derivatives and Drug Conjugates Thereof to the Folate Receptor-Reference-Cited by-同舟云学术

Properties Influencing the Relative Binding Affinity of Pteroate Derivatives and Drug Conjugates Thereof to the Folate Receptor

Published:2009-02-03 Issue:6 Volume:26 Page:1315-1323
ISSN:0724-8741
Container-title:Pharmaceutical Research
language:en
Short-container-title:Pharm Res

Author:

Leamon Christopher P.,You Fei,Santhapuram Hari Krishna,Fan Mingjin,Vlahov Iontcho R.

Publisher

Springer Science and Business Media LLC

Subject

Pharmacology (medical),Organic Chemistry,Pharmaceutical Science,Pharmacology,Molecular Medicine,Biotechnology

Link

http://link.springer.com/content/pdf/10.1007/s11095-009-9840-3.pdf

Reference25 articles.

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2. C. P. Leamon, and P. S. Low. Membrane folate-binding proteins are responsible for folate- protein conjugate endocytosis into cultured cells. Biochem. J. 291:855–860 (1993).

3. I. G. Campbell, T. A. Jones, W. D. Foulkes, and J. Trowsdale. Folate-binding protein is a marker for ovarian cancer. Cancer Res. 51:5329–5338 (1991).

4. C. P. Leamon, and J. A. Reddy. Folate-targeted chemotherapy. Adv. Drug Deliv. Rev. 56:1127–1141 (2004) doi: 10.1016/j.addr.2004.01.008 .

5. J. A. Reddy, R. Dorton, E. Westrick, A. Dawson, T. Smith, L. C. Xu, M. Vetzel, P. Kleindl, I. R. Vlahov, and C. P. Leamon. Preclinical evaluation of EC145, a folate-Vinca alkaloid conjugate. Cancer Res. 67:4434–4442 (2007) doi: 10.1158/0008-5472.CAN-07-0033 .

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