Projecting ADME Behavior and Drug-Drug Interactions in Early Discovery and Development: Application of the Extended Clearance Classification System

Author:

El-Kattan Ayman F.,Varma Manthena V.,Steyn Stefan J.,Scott Dennis O.,Maurer Tristan S.,Bergman Arthur

Publisher

Springer Science and Business Media LLC

Subject

Pharmacology (medical),Organic Chemistry,Pharmaceutical Science,Pharmacology,Molecular Medicine,Biotechnology

Reference58 articles.

1. Beaumont K, Smith DA. Does human pharmacokinetic prediction add significant value to compound selection in drug discovery research? Curr Opin Drug Discov Devel. 2009;12(1):61–71.

2. Mager DE. Quantitative structure-pharmacokinetic/pharmacodynamic relationships. Adv Drug Deliv Rev. 2006;58(12–13):1326–56.

3. Rostami-Hodjegan A, Tucker GT. Simulation and prediction of in vivo drug metabolism in human populations from in vitro data. Nat Rev. 2007;6(2):140–8.

4. van de Waterbeemd H, Gifford E. ADMET in silico modelling: towards prediction paradise? Nat Rev. 2003;2(3):192–204.

5. van De Waterbeemd H, Smith DA, Beaumont K, Walker DK. Property-based design: optimization of drug absorption and pharmacokinetics. J Med Chem. 2001;44(9):1313–33.

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