Novel approach of multi-targeted thiazoles and thiazolidenes toward anti-inflammatory and anticancer therapy—dual inhibition of COX-2 and 5-LOX enzymes-Reference-Cited by-同舟云学术

Novel approach of multi-targeted thiazoles and thiazolidenes toward anti-inflammatory and anticancer therapy—dual inhibition of COX-2 and 5-LOX enzymes

Published:2020-11-01 Issue:1 Volume:30 Page:236-257
ISSN:1054-2523
Container-title:Medicinal Chemistry Research
language:en
Short-container-title:Med Chem Res

Author:

P Jaismy Jacob,S L Manju

Publisher

Springer Science and Business Media LLC

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics

Link

http://link.springer.com/content/pdf/10.1007/s00044-020-02655-9.pdf

Reference53 articles.

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3. Mantovani A, Allavena P, Sica A, Balkwill F. Cancer-related inflammation. Nature. 2008;54:436. https://doi.org/10.1038/nature07205.

4. Manju SL, Ethiraj KR, Elias G. Safer anti-inflammatory therapy through dual COX-2/5-LOX inhibitors: a structure-based approach. Eur J Pharm Sci. 2018;121:356–381. https://doi.org/10.1016/j.ejps.2018.06.003.

5. Singh P, Kaur J, Singh G, Bhatti R. Triblock conjugates: identification of a highly potent antiinflammatory agent. J Med Chem. 2015;58:5989–6001. https://doi.org/10.1021/acs.jmedchem.5b00952.

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