Structural insights into mode of actions of novel substituted 4- and 6-azaindole-3-carboxamides analogs as renin inhibitors: molecular modeling studies

Author:

Sharma Mukesh C.

Publisher

Springer Science and Business Media LLC

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics

Reference103 articles.

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3. Bhadoriya KS, Kumawat NK, Bhavthankar SV, Avchar MA, Dhuma DM, Patil SD, Jain SV (2012) Exploring 2D and 3D QSARs of benzimidazole derivatives as transient receptor potential melastatin (TRPM8) antagonists using MLR and kNN-MFA methodology. J Saudi Chem Soc. doi: 10.1016/j.jscs.2012.11.001

4. Bhadoriya KS, Sharma MC, Sharma S, Jain SV, Avchar MH (2013a) An approach to design potent anti-Alzheimer’s agents by 3D QSAR studies on fused 5,6-bicyclic heterocycles as c-secretase modulators using kNN-MFA methodology. Arab J Chem. doi: 10.1016/j.arabjc.2013.02.002

5. Bhadoriya KS, Sharma MC, Jain SV, Raut GS, Rananaware JR (2013b) Three-dimensional quantitative structure–activity relationship (3D-QSAR) analysis and molecular docking-based combined in silico rational approach to design potent and novel TRPV1 antagonists. Med Chem Res 22:2312–2327

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