Study on structure-activity relationship (SAR) of simplified mirogabalin derivatives as voltage-gated calcium channel α2δ ligands for the treatment of chronic neuropathic pain-Reference-Cited by-同舟云学术

Study on structure-activity relationship (SAR) of simplified mirogabalin derivatives as voltage-gated calcium channel α2δ ligands for the treatment of chronic neuropathic pain

Published:2022-12-26 Issue:2 Volume:32 Page:288-313
ISSN:1054-2523
Container-title:Medicinal Chemistry Research
language:en
Short-container-title:Med Chem Res

Author:

Zhang Yuanwen,Zheng Yueming,Wu Qingqing,Tian Fuyun,Ma Chuanjun,Xu Haiyan,Zhan Li,Gao Zhaobing^ORCID,Zhao Guilong^ORCID,Ti Huihui^ORCID

Funder

Basic and Applied Basic Research Foundation of Guangdong Province

Zhongshan Science and Technology Bureau

Guangdong Provincial High-Level New R&D Institute Strategic Special Fund

Special Fund for Scientific Innovation Strategy-Construction of High-level Academy of Agriculture Science

National Natural Science Foundation of China

Publisher

Springer Science and Business Media LLC

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics

Link

https://link.springer.com/content/pdf/10.1007/s00044-022-03006-6.pdf

Reference36 articles.

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3. Shinu P, Morsy MA, Nair AB, Al Mouslem AK, Venugopala KN, Goyal M, et al. Novel therapies for the treatment of neuropathic pain: potential and pitfalls. J Clin Med. 2022;11:3002. https://doi.org/10.3390/jcm11113002.

4. Inoue S, Taguchi T, Yamashita T, Nakamura M, Ushida T. The prevalence and impact of chronic neuropathic pain on daily and social life: a nationwide study in a Japanese population. Eur J Pain. 2017;21:727–37. https://doi.org/10.1002/ejp.977.

5. Stefano GD, Lionardo AD, Pietro GD, Cruccu G, Truini A. Pharmacotherapeutic options for managing neuropathic pain: a systematic review and meta-analysis. Pain Res Manag. 2021:6656863. https://doi.org/10.1155/2021/6656863.

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