Docking studies of some 5-hydroxypyridine-4-one derivatives: evaluation of integrase and ribonuclease H domain of reverse transcriptase as possible targets for anti-HIV-1 activity-Reference-Cited by-同舟云学术

Docking studies of some 5-hydroxypyridine-4-one derivatives: evaluation of integrase and ribonuclease H domain of reverse transcriptase as possible targets for anti-HIV-1 activity

Published:2014-11-06 Issue:5 Volume:24 Page:2195-2212
ISSN:1054-2523
Container-title:Medicinal Chemistry Research
language:en
Short-container-title:Med Chem Res

Author:

Sirous Hajar,Zabihollahi Rezvan,Aghasadeghi Mohammad R.,Sadat Seyed Mehdi,Saghaie Lotfollah,Fassihi Afshin

Publisher

Springer Science and Business Media LLC

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics

Link

http://link.springer.com/content/pdf/10.1007/s00044-014-1289-1.pdf

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4. Barré-Sinoussi F, Chermann JC, Rey F, Nugeyre MT, Chamaret S, Gruest J, Dauguet C, Axler-Blin C, Vezinet-Brun F, Rouzioux C, Rozenbaum W, Mon-tagnier L (1983) Isolation of a T-lymphotropic retrovirus from a patient at risk for acquired immune deficiency syndrome (AIDS). Science 220:868–871

5. Budihas S, Gorshkova I, Gaidamakov S, Wamiru A, Bona M, Parniak M, Crouch R, McMahon J, Beutler J, Le Grice S (2005) Selective inhibition of HIV-1 reverse transcriptase-associated ribonu-clease H activity by hydroxylated tropolones. Nucleic Acids Res 33:1249–1256

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