Evaluation of 3-carbamoylpropanoic acid analogs as inhibitors of human hypoxia-inducible factor (HIF) prolyl hydroxylase domain enzymes
Author:
Funder
Research University Grant
Publisher
Springer Science and Business Media LLC
Subject
Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics
Link
http://link.springer.com/content/pdf/10.1007/s00044-020-02681-7.pdf
Reference46 articles.
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3. Semenza GL. “Oxygen-regulated transcription factors and their role in pulmonary disease.”. Respir Res. 2000;1:159–62.
4. Epstein Andrew CR, et al. C. Elegans EGL-9 and mammalian homologs define a family of dioxygenases that regulate hif by prolyl hydroxylation. Cell. 2001;107:43–54.
5. Chowdhury R, et al. Structural basis for oxygen degradation domain selectivity of the hif prolyl hydroxylases. Nat Commun. 2016;7:12673.
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