Novel Benzo[4,5]imidazo[1,2-a]pyrimidine derivatives as selective Cyclooxygenase-2 Inhibitors: Design, synthesis, docking studies, and biological evaluation-Reference-Cited by-同舟云学术

Novel Benzo[4,5]imidazo[1,2-a]pyrimidine derivatives as selective Cyclooxygenase-2 Inhibitors: Design, synthesis, docking studies, and biological evaluation

Published:2023-01-23 Issue:3 Volume:32 Page:495-505
ISSN:1054-2523
Container-title:Medicinal Chemistry Research
language:en
Short-container-title:Med Chem Res

Author:

Bayanati Maryam,Khoramjouy Mona,Faizi Mehrdad,Movahed Mahsa Azami,Mahboubi-Rabbani Mohammad,Zarghi Afshin

Publisher

Springer Science and Business Media LLC

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics

Link

https://link.springer.com/content/pdf/10.1007/s00044-023-03022-0.pdf

Reference44 articles.

1. Khare A, Trivedi S, Rajak H, Pawar R, Patil U, Singour P. Hansch analysis of novel pyrimidine derivatives as highly potent and specific COX-2 inhibitors. Med Chem Res. 2012;21:672–80. https://doi.org/10.1007/s00044-011-9566-8

2. Zarghi A, Arfaei S. Selective COX-2 inhibitors: a review of their structure-activity relationships. Iran J Pharm Res. 2011;10:655. https://doi.org/10.22037/ijpr.2011.1047

3. Makar KW, Poole EM, Resler AJ, Seufert B, Curtin K, Kleinstein SE, et al. COX-1 (PTGS1) and COX-2 (PTGS2) polymorphisms, NSAID interactions, and risk of colon and rectal cancers in two independent populations. Cancer Causes Control. 2013;24:2059–75. https://doi.org/10.1007/s10552-013-0282-1

4. Willoughby DA, Moore AR, Colville-Nash PR. COX-1, COX-2, and COX-3 and the future treatment of chronic inflammatory disease. Lancet. 2000;355:646–8. https://doi.org/10.1016/S0140-6736(99)12031-2

5. Vane JR, Botting RM. Mechanism of action of nonsteroidal anti-inflammatory drugs. Am J Med. 1998;104:2S–8S. https://doi.org/10.1016/S0002-9343(97)00203-9

Cited by 8 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Novel 3-substituted coumarins inspire a custom pharmacology prediction pipeline: an anticancer discovery adventure;Future Medicinal Chemistry;2024-09-04

2. Selective COX-2 inhibitors as anticancer agents: a patent review (2018-2023);Expert Opinion on Therapeutic Patents;2024-07-03

3. Conjugate and regiochemical addition of aminoazoles to 2-(4-(2,2-dicyanovinyl)phenoxy)-N-arylacetamide affording fused pyrimidines linked to phenoxy-N-arylacetamide: Antibacterial activity, molecular docking, and DNA binding studies;Journal of Molecular Structure;2024-07

4. Design, Synthesis, In vitro and In vivo Evaluation of New Imidazo[1,2-a]pyridine Derivatives as Cyclooxygenase-2 Inhibitors;Anti-Cancer Agents in Medicinal Chemistry;2024-04

5. Reaction of 2-Aminobenzimidazoles with Acetylene in the KOBut/DMSO System. Self-Assembly of Benzo[d]imidazo[1,2-a]imidazoles and Benzo[4,5]imidazo[1,2-a]pyrimidines under Competition between Nucleophilic Centers;Russian Journal of Organic Chemistry;2024-02