Benzenesulfonamides bearing pyrrolidinone moiety as inhibitors of carbonic anhydrase IX: synthesis and binding studies
Author:
Funder
Research Council of Lithuania
Publisher
Springer Science and Business Media LLC
Subject
Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics
Link
http://link.springer.com/content/pdf/10.1007/s00044-016-1741-5.pdf
Reference32 articles.
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2. Aspatwar A, Tolvanen ME, Ortutay C, Parkkila S (2014) Carbonic anhydrase related proteins: molecular biology and evolution. Subcell Biochem 75:135–156
3. Baranauskienė L, Hilvo M, Matulienė J, Golovenko D, Manakova E, Dudutienė V, Michailovienė V, Torresan J, Jachno J, Parkilla S, Maresca A, Supuran CT, Gražulis S, Matulis D (2010) Inhibition and binding studies of carbonic anhydrase isozymes I,II and IX with benzimidazo[1,2c][1,2,3]thiadiazole-7-sulphonamides. J Enzyme Inhib Med Chem 25:863–870
4. Cimmperman P, Baranauskienė L, Jachimovičiūtė S, Jachno J, Torresan J, Michailovienė V, Matulienė J, Sereikaitė J, Bumelis V, Matulis D (2008) A quantitative model of thermal stabilization and destabilization of proteins by ligands. Biophys J 95:3222–3231
5. Dudutienė V, Matulienė J, Smirnov A, Timm DD, Zubrienė A, Baranauskienė L, Morkūnaitė V et al. (2014) Discovery and characterization of novel selective inhibitors of carbonic anhydrase IX. J Med Chem 57:9435–9446
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