The importance of tamoxifen metabolism in tamoxifen-stimulated breast tumor growth

Author:

Osborne C. Kent,Jarman Michael,McCague Ray,Coronado Ester B.,Hilsenbeck Susan G.,Wakeling Alan E.

Publisher

Springer Science and Business Media LLC

Subject

Pharmacology (medical),Cancer Research,Pharmacology,Toxicology,Oncology

Reference22 articles.

1. Buckley MM, Goa KL (1989) Tamoxifen: a reappraisal of its pharmacodynamic and pharmacokinetic properties and therapeutic use. Drugs 37: 451?490

2. Dowsett M, Johnston SRD, Haynes BP, Sacks NPM, Baum MB, Ebbs SR, Smith IE (1993) Impaired intra-tumoral uptake of tamoxifen as a mechanism for resistance in human breast cancer. Proc Am Assoc Cancer Res 34: 1463A

3. Early Breast Cancer Trialists Collaborative Group (1992) Systemic treatment of early breast cancer by hormonal, systemic or immune therapy: 133 randomized trials involving 31,000 recurrences and 24,000 deaths among 75,000 women. Lancet 339: 1?15, 71?85

4. Encarnacion CA, Ciocca DR, McGuire WL, Clark GM, Fuqua SAW, Osborne CK (1993) Measurement of steroid hormone receptors in breast cancer patients on tamoxifen. Breast Cancer Res Treat 26: 237?246

5. Gottardis MM, Jordan VC (1988) Development of tamoxifen-stimulated growth of MCF-7 tumors in athymic mice after long-term antiestrogen administration. Cancer Res 48: 5183?5187

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