Radiosynthesis and in vivo evaluation of a series of substituted 11C-phenethylamines as 5-HT2A agonist PET tracers-Reference-Cited by-同舟云学术

Radiosynthesis and in vivo evaluation of a series of substituted 11C-phenethylamines as 5-HT2A agonist PET tracers

Published:2010-12-21 Issue:4 Volume:38 Page:681-693
ISSN:1619-7070
Container-title:European Journal of Nuclear Medicine and Molecular Imaging
language:en
Short-container-title:Eur J Nucl Med Mol Imaging

Author:

Ettrup Anders,Hansen Martin,Santini Martin A.,Paine James,Gillings Nic,Palner Mikael,Lehel Szabolcs,Herth Matthias M.,Madsen Jacob,Kristensen Jesper,Begtrup Mikael,Knudsen Gitte M.

Publisher

Springer Science and Business Media LLC

Subject

Radiology Nuclear Medicine and imaging,General Medicine,Radiology Nuclear Medicine and imaging,General Medicine

Link

http://link.springer.com/content/pdf/10.1007/s00259-010-1686-8.pdf

Reference31 articles.

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3. Pinborg LH, Adams KH, Svarer C, et al. Quantification of 5-HT2A receptors in the human brain using [18F]altanserin-PET and the bolus/infusion approach. J Cereb Blood Flow Metab. 2003;23:985–96.

4. Ito H, Nyberg S, Halldin C, Lundkvist C, Farde L. PET imaging of central 5-HT2A receptors with carbon-11-MDL 100,907. J Nucl Med. 1998;39:208–14.

5. Fitzgerald LW, Conklin DS, Krause CM, et al. High-affinity agonist binding correlates with efficacy (intrinsic activity) at the human serotonin 5-HT2A and 5-HT2C receptors: evidence favoring the ternary complex and two-state models of agonist action. J Neurochem. 1999;72:2127–34.

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