Interspecies differences in plasma protein binding of MS-275, a novel histone deacetylase inhibitor

Author:

Acharya Milin R.,Sparreboom Alex,Sausville Edward A.,Conley Barbara A.,Doroshow James H.,Venitz Jűrgen,Figg William D.

Publisher

Springer Science and Business Media LLC

Subject

Pharmacology (medical),Cancer Research,Pharmacology,Toxicology,Oncology

Reference18 articles.

1. Acharya MR, Baker SD, Verweij J, Figg WD, Sparreboom A (2004) Determination of fraction unbound docetaxel using micro-equilibrium dialysis. Anal Biochem 331:192

2. Bacchus H (1975) Serum glycoproteins in cancer. Prog Clin Pathol 6:111

3. Benet LZ, Hoener BA (2002) Changes in plasma protein binding have little clinical relevance. Clin Pharmacol Ther 71:115

4. Dasgupta A (2002) Clinical utility of free drug monitoring. Clin Chem Lab Med 40:986

5. Fuse E, Tanii H, Kurata N, Kobayashi H, Shimada Y, Tamura T, Sasaki Y, Tanigawara Y, Lush RD, Headlee D, Figg WD, Arbuck SG, Senderowicz AM, Sausville EA, Akinaga S, Kuwabara T, Kobayashi S (1998) Unpredicted clinical pharmacology of UCN-01 caused by specific binding to human alpha1-acid glycoprotein. Cancer Res 58:3248

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