Metabolism of diazepam and related benzodiazepines by human liver microsomes

Author:

Hooper W. D.,Watt J. A.,Mckinnon G. E.,Reelly P. E. B.

Publisher

Springer Science and Business Media LLC

Subject

Pharmacology (medical),Pharmacology

Reference38 articles.

1. Stembach L.H. (1973): Chemistry of 1,4-benzodiazepines and some aspects of the structure-activity-relationship. In: Garattini S., Mussini E., Randall L.O. (eds). The Benzodiazepines. New York, Raven Press, pp. 1–26.

2. Schwartz M.A. (1973): Pathways of metabolism of the benzodiazepines. In: Garattini S., Mussini E., Randall L.O. (eds). The Benzodiazepines. New York, Raven Press, pp. 53–74.

3. Garattini S., Mussini E., Marcucci F., Guaitani A. (1973): Metabolic studies on benzodiazepines. In: Garattini S., Mussini E., Randall L.O. (eds). The Benzodiazepines. New York, Raven Press, pp. 75–97.

4. Mussini E., Marcucci F., Fanelli R., Garattini S. (1971): Metabolism of diazepam and its metabolites by guinea pig liver microsomes. Biochem. Pharmacol., 20, 2529–2531.

5. Lu X.-L., Yang S.K. (1989): Metabolism of prazepam by rat liver microsomes: stereoselective formation and tf-dealkylation of 3-hydroxyprazepam. Mol. Pharmacol., 36, 932–938.

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