De novo design of VEGFR-2 tyrosine kinase inhibitors based on a linked-fragment approach

Author:

Liu Yi-zhou,Wang Xiao-li,Wang Xin-ying,Yu Ri-lei,Liu Dong-qing,Kang Cong-min

Funder

National Natural Science Foundation of China

Fundamental Research Funds for the Central Universities

Publisher

Springer Science and Business Media LLC

Subject

Computational Theory and Mathematics,Inorganic Chemistry,Organic Chemistry,Physical and Theoretical Chemistry,Computer Science Applications,Catalysis

Reference34 articles.

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3. Steri V, Ellison TS, Gontarczyk AM, Weilbaecher K, Schneider JG, Edwards D, Fruttiger M, Hodivala-Dilke KM, Robinson SD (2014) Acute depletion of endothelial β3-integrin transiently inhibits tumor growth and angiogenesis in mice. Circ Res 114:79–91

4. Deng YH, Xu D, Su YX, Cheng YJ, Yang YL, Wang XY, Zhang J, You QD, Sun LP (2015) Synthesis and biological evaluation of novel oxazolo [5, 4‐d] pyrimidines as potent VEGFR‐2 inhibitors. Chem Biodivers 12:528–537

5. Takahashi Y, Kitadai Y, Bucana CD, Cleary KR, Ellis LM (1995) Expression of vascular endothelial growth factor and its receptor, KDR, correlates with vascularity, metastasis, and proliferation of human colon cancer. Cancer Res 55:3964–3968

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