1. Burger A (1991) Isosterism and bioisosterism in drug design. Progress Drug Res 37:288–362
2. Patani GA, LaVoie EJ (1996) Bioisosterism: a rational approach in drug design. Chem Rev 96:3147–3176
3. Thornber CW (1979) Isosterism and molecular modification in drug design. Chem Soc Rev 8:563–580
4. Lipinski CA (1986) Bioisosterism in drug design. Ann Rep Med Chem 21:283–291
5. Wermuth CG, Bourguignon J-J (2003) In: Wermuth CG (ed) The practice of medicinal chemistry, 2nd edn. Chaps 12–16, Academic, London, pp 181–310. ISBN: 0-12-744640-0