Development of Non-GAT1-Selective Inhibitors: Challenges and Achievements-Reference-Cited by-同舟云学术

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Development of Non-GAT1-Selective Inhibitors: Challenges and Achievements

Published:2017 Issue: Volume: Page:315-332
ISSN:2190-5215
Container-title:Advances in Neurobiology
language:
Short-container-title:

Author:

Damgaard Maria,Haugaard Anne Stæhr,Kickinger Stefanie,Al-Khawaja Anas,Lie Maria E. K.,Ecker Gerhard F.,Clausen Rasmus Prætorius,Frølund Bente

Publisher

Springer International Publishing

Link

http://link.springer.com/content/pdf/10.1007/978-3-319-55769-4_16

Reference65 articles.

1. Al-Khawaja A, Petersen JG, Damgaard M, Jensen MH, Vogensen SB, Lie ME, et al. Pharmacological identification of a guanidine-containing β-alanine analogue with low micromolar potency and selectivity for the betaine/GABA transporter 1 (BGT1). Neurochem Res. 2014;39(10):1988–96.

2. Alexander SP, Kelly E, Marrion N, Peters JA, Benson HE, Faccenda E, et al. The concise guide to pharmacology 2015/16: transporters. Br J Pharmacol. 2015;172(24):6110–202.

3. Ali FE, Bondinell WE, Dandridge PA, Frazee JS, Garvey E, Girard GR, et al. Orally active and potent inhibitors of gamma-aminobutyric acid uptake. J Med Chem. 1985;28(5):653–60.

4. Baglo Y, Gabrielsen M, Sylte I, Gederaas OA. Homology modeling of human gamma-butyric acid transporters and the binding of pro-drugs 5-aminolevulinic acid and methyl aminolevulinic acid used in photodynamic therapy. PLoS One. 2013;8(6):e65200.

5. Beuming T, Shi L, Javitch JA, Weinstein H. A comprehensive structure-based alignment of prokaryotic and eukaryotic neurotransmitter/Na+ symporters (NSS) aids in the use of the LeuT structure to probe NSS structure and function. Mol Pharmacol. 2006;70(5):1630–42.

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