Unravelling the Structural Mechanism of Action of 5-methyl-5-[4-(4-oxo-3H-quinazolin-2-yl)phenyl]imidazolidine-2,4-dione in Dual-Targeting Tankyrase 1 and 2: A Novel Avenue in Cancer Therapy-Reference-Cited by-同舟云学术

Unravelling the Structural Mechanism of Action of 5-methyl-5-[4-(4-oxo-3H-quinazolin-2-yl)phenyl]imidazolidine-2,4-dione in Dual-Targeting Tankyrase 1 and 2: A Novel Avenue in Cancer Therapy

Published:2022-05-30 Issue:3 Volume:80 Page:505-518
ISSN:1085-9195
Container-title:Cell Biochemistry and Biophysics
language:en
Short-container-title:Cell Biochem Biophys

Author:

Peters Xylia Q.,Agoni Clement,Soliman Mahmoud E. S.

Publisher

Springer Science and Business Media LLC

Subject

Cell Biology,Biochemistry,General Medicine,Biophysics

Link

https://link.springer.com/content/pdf/10.1007/s12013-022-01076-2.pdf

Reference71 articles.

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2. Haikarainen, T., Koivunen, J., Narwal, M., Venkannagari, H., Obaji, E., Joensuu, P., & Lehtiö, L. (2013). Para-substituted 5-methyl-5-[4-(4-oxo-3H-quinazolin-2-yl)phenyl]imidazolidine-2,4-diones as potent and selective tankyrase inhibitors. ChemMedChem, 8(12), 1978–1985. https://doi.org/10.1002/cmdc.201300337.

3. Peters, X. Q., Malinga, T. H., Agoni, C., Olotu, F. A., & Soliman, M. E. S. (2019). Zoning in on Tankyrases: a brief review on the past, present and prospective studies. Anti-Cancer Agents in Medicinal Chemistry, 19(16), 1920–1934. https://doi.org/10.2174/1871520619666191019114321.

4. Verma, A., Kumar, A., Chugh, A., Kumar, S. & Kumar, P. (2020). Tankyrase inhibitors: emerging and promising therapeutics for cancer treatment. Medicinal Chemistry Research, 30(1), 50–73. https://doi.org/10.1007/S00044-020-02657-7.

5. Ferri, M., Liscio, P., Carotti, A., Asciutti, S., Sardella, R., Macchiarulo, A., & Camaioni, E. (2017). Targeting Wnt-driven cancers: discovery of novel tankyrase inhibitors. European Journal of Medicinal Chemistry. https://doi.org/10.1016/j.ejmech.2017.09.030.

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