Synthesis and anti-inflammatory evaluation of new 1,3,5-triaryl-4,5-dihydro-1H-pyrazole derivatives possessing an aminosulphonyl pharmacophore-Reference-Cited by-同舟云学术

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Synthesis and anti-inflammatory evaluation of new 1,3,5-triaryl-4,5-dihydro-1H-pyrazole derivatives possessing an aminosulphonyl pharmacophore

Published:2015-04-23 Issue:11 Volume:38 Page:1932-1942
ISSN:0253-6269
Container-title:Archives of Pharmacal Research
language:en
Short-container-title:Arch. Pharm. Res.

Author:

Abdellatif Khaled R. A.,Abdelgawad Mohamed A.,Elshemy Heba A. H.,Alsayed Shahinda S. R.,Kamel Gehan

Publisher

Springer Science and Business Media LLC

Subject

Organic Chemistry,Drug Discovery,Molecular Medicine

Link

http://link.springer.com/content/pdf/10.1007/s12272-015-0606-7.pdf

Reference36 articles.

1. Abdelazeem, A.H., S.A. Abdelatef, M.T. El-Saadi, H.A. Omar, S.I. Khan, C.R. McCurdy, and S.M. El-Moghazy. 2014. Novel pyrazolopyrimidine derivatives targeting COXs and iNOS enzymes; design, synthesis and biological evaluation as potential anti-inflammatory agents. European Journal of Pharmaceutical Sciences 62: 197–211.

2. Abdellatif, K.R.A., M.A. Chowdhury, and E.E. Knaus. 2008a. Synthesis of new 1-[4-methane (amino) sulfonylphenyl)]-5-[4- (aminophenyl)]-3-trifluoromethyl-1H-pyrazoles. Journal of Heterocyclic Chemistry 45: 1707–1710.

3. Abdellatif, K.R.A., M.A. Chowdhury, C.A. Velázquez, Z. Huang, Y. Dong, D. Das, G. Yu, M.R. Suresh, and E.E. Knaus. 2010. Celecoxib prodrugs possessing a diazen-1-ium-1,2-diolate nitric oxide donor moiety: synthesis, biological evaluation and nitric oxide release studies. Bioorganic & Medicinal Chemistry Letters 20: 4544–4549.

4. Abdellatif, K.R.A., M.A. Chowdhury, Y. Dong, D. Das, G. Yu, C. Velázquez, M.R. Suresh, and E.E. Knaus. 2009. Diazen-1-ium-1,2-diolated nitric oxide donor ester prodrugs of 5-(4-carboxymethylphenyl)-1-(4-methanesulfonylphenyl)-3-trifluoromethyl-1H-pyrazole and its aminosulfonyl analog: Synthesis, biological evaluation and nitric oxide release studies. Bioorganic & medicinal chemistry 17: 5182–5188.

5. Abdellatif, K.R.A., M.A. Chowdhury, Y. Dong, and E.E. Knaus. 2008b. Diazen-1-ium-1,2-diolated nitric oxide donor ester prodrugs of 1-(4-methanesulfonylphenyl)-5-aryl-1H-pyrazol-3-carboxylic acids: synthesis, nitric oxide release studies and anti-inflammatory activities. Bioorganic & medicinal chemistry 16: 6528–6534.

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