Structure–activity relationships of novel quinazoline derivatives with high selectivity for HER2 over EGFR
Author:
Funder
Ministry of Education
Publisher
Springer Science and Business Media LLC
Subject
Organic Chemistry,Drug Discovery,Molecular Medicine
Link
https://link.springer.com/content/pdf/10.1007/s12272-022-01376-4.pdf
Reference17 articles.
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3. Arteaga CL, O’Neill A, Moulder SL, Pins M, Sparano JA, Sledge GW, Davidson NE (2008) A phase I–II study of combined blockade of the ErbB receptor network with trastuzumab and gefitinib in patients with HER2 (ErbB2)-overexpressing metastatic breast cancer. Clin Cancer Res 14:6277–6283. https://doi.org/10.1158/1078-0432.CCR-08-0482
4. Baselga J, Coleman RE, Cortés J, Janni W (2017) Advances in the management of HER2-positive early breast cancer. Crit Rev Oncol Hematol 119:113–122. https://doi.org/10.1016/j.critrevonc.2017.10.001
5. Buonomo OC, Caredda E, Portarena I, Vanni G, Orlandi A, Bagni C, Petrella G, Palombi L, Orsaria P (2017) New insights into the metastatic behavior after breast cancer surgery, according to well-established clinicopathological variables and molecular subtypes. PLoS ONE 12:e0184680. https://doi.org/10.1371/journal.pone.0184680
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