Fluorinated pyrrole incorporated 2-thiazolyl hydrazone motifs: a new class of antimicrobial and anti tuberculosis agents

Author:

Sowmya P. V.,Poojary Boja,Kumar Vasantha,Vishwanatha U.,Shetty Premalatha

Publisher

Springer Science and Business Media LLC

Subject

Organic Chemistry,Drug Discovery,Molecular Medicine

Reference40 articles.

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3. Battilocchio C, Poce G, Alfonso S, Porretta GC, Consalvi S, Sautebin L, Pace S, Rossi A, Ghelardini C, Mannelli LDC, Schenone S, Giordani A, Francesco LD, Patrignani P, Biava M (2013) A class of pyrrole derivatives endowed with analgesic/antiinflammatory activity. Bioorg Med Chem 21:3695–3701

4. Bell FW, Cantrell AS, Hogberg M, Jaskunas SR, Johansson NG, Jordon CL, Kinnick MD, Lind P, Morin JM, Noreen R, Oberg B, Palkowitz JA, Parrish CA, Pranc P, Sahlberg C, Ternansky RJ, Vasileff RT, Vrang L, West SJ, Zhang H, Zhou XX (1995) Phenethylthiazolethiourea (PETT) compounds, a new class of HIV-1 reverse transcriptase inhibitors 1. Synthesis and basic structure-activity relationship studies of PETT analogs. J Med Chem 38:4929–4936

5. Biava M, Porretta GC, Poce G, Logu AD, Meleddu R, Rossi ED, Manetti F, Botta M (2009) 1,5-Diaryl-2-ethyl pyrrole derivatives as antimycobacterial agents: design, synthesis, and microbiological evaluation. Eur J Med Chem 44:4734–4738

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