A convenient one-pot synthesis of novel heterocyclic systems of 9-chloro-4-methyl-6,11-dihydro-5H-benzo[b]pyrimido[4,5-e][1,4]diazepine and inhibitory evaluation against bromodomain-containing protein 4 (BRD4) enzyme by molecular docking-Reference-Cited by-同舟云学术

A convenient one-pot synthesis of novel heterocyclic systems of 9-chloro-4-methyl-6,11-dihydro-5H-benzo[b]pyrimido[4,5-e][1,4]diazepine and inhibitory evaluation against bromodomain-containing protein 4 (BRD4) enzyme by molecular docking

Published:2023-09-14 Issue:11 Volume:20 Page:2841-2848
ISSN:1735-207X
Container-title:Journal of the Iranian Chemical Society
language:en
Short-container-title:J IRAN CHEM SOC

Author:

Assadzadeh Fahimeh,Afrough Toktam,Eshghi Hossein^ORCID,Sabet-Sarvestani Hossein

Publisher

Springer Science and Business Media LLC

Subject

General Chemistry

Link

https://link.springer.com/content/pdf/10.1007/s13738-023-02880-0.pdf

Reference30 articles.

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4. E.Y. Zelina et al., A Route to (Het) arene-annulated pyrrolo [1, 2-d][1, 4] diazepines via the expanded intramolecular paal-knorr reaction: nitro group and furan ring as equivalents of amino group and 1, 4-diketone. J. Org. Chem. 84(21), 13707–13720 (2019). https://doi.org/10.1021/acs.joc.9b01925

5. H. Farhid et al., Multicomponent reactions as a potent tool for the synthesis of benzodiazepines. Org. Biomol. Chem. (2021). https://doi.org/10.1039/D0OB02600J