Correlations between metabolism and structural elements of the alicyclic fentanyl analogs cyclopropyl fentanyl, cyclobutyl fentanyl, cyclopentyl fentanyl, cyclohexyl fentanyl and 2,2,3,3-tetramethylcyclopropyl fentanyl studied by human hepatocytes and LC-QTOF-MS-Reference-Cited by-同舟云学术

Correlations between metabolism and structural elements of the alicyclic fentanyl analogs cyclopropyl fentanyl, cyclobutyl fentanyl, cyclopentyl fentanyl, cyclohexyl fentanyl and 2,2,3,3-tetramethylcyclopropyl fentanyl studied by human hepatocytes and LC-QTOF-MS

Published:2018-10-25 Issue:1 Volume:93 Page:95-106
ISSN:0340-5761
Container-title:Archives of Toxicology
language:en
Short-container-title:Arch Toxicol

Author:

Åstrand Anna^ORCID,Töreskog Amanda,Watanabe Shimpei^ORCID,Kronstrand Robert^ORCID,Gréen Henrik^ORCID,Vikingsson Svante^ORCID

Funder

VINNOVA

Strategic Research Area in Forensic Science

Publisher

Springer Science and Business Media LLC

Subject

Health, Toxicology and Mutagenesis,Toxicology,General Medicine

Link

http://link.springer.com/article/10.1007/s00204-018-2330-9/fulltext.html

Reference22 articles.

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2. Drug Enforcement Administration DoJ (2018a) Schedules of controlled substances: temporary placement of cyclopropyl fentanyl in schedule I. Temporary amendment; temporary scheduling order. Fed Regist 83(3):469–472

3. Drug Enforcement Administration DoJ (2018b) Schedules of controlled substances: temporary placement of seven fentanyl-related substances in schedule I. Fed Regist 83(22):4880–4885

4. EMCDDA (2017a) Report on the risk assessment of N-(1–phenethylpiperidin-4-yl)-N-phenylacrylamide (acryloylfentanyl) in the framework of the Council Decision on new psychoactive substances. EMCDDA, Lisbon

5. EMCDDA (2017b) Report on the risk assessment of N-phenyl-N-[1-(2-phenylethyl)piperidin-4-yl]furan-2-carboxamide (furanylfentanyl) in the framework of the Council Decision on new psychoactive substances. EMCDDA, Lisbon

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