In silico, in vitro, and in vivo human metabolism of acetazolamide, a carbonic anhydrase inhibitor and common “diuretic and masking agent” in doping-Reference-Cited by-同舟云学术

In silico, in vitro, and in vivo human metabolism of acetazolamide, a carbonic anhydrase inhibitor and common “diuretic and masking agent” in doping

Published:2022-04-11 Issue:7 Volume:96 Page:1989-2001
ISSN:0340-5761
Container-title:Archives of Toxicology
language:en
Short-container-title:Arch Toxicol

Author:

Busardò Francesco P.^ORCID,Lo Faro Alfredo F.^ORCID,Sirignano Ascanio^ORCID,Giorgetti Raffaele^ORCID,Carlier Jeremy^ORCID

Funder

Ministero della Salute

Publisher

Springer Science and Business Media LLC

Subject

Health, Toxicology and Mutagenesis,Toxicology,General Medicine

Link

https://link.springer.com/content/pdf/10.1007/s00204-022-03289-z.pdf

Reference57 articles.

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3. Carlier J, Diao X, Scheidweiler KB, Huestis MA (2017) Distinguishing intake of new synthetic cannabinoids ADB-PINACA and 5F-ADB-PINACA with human hepatocyte metabolites and high-resolution mass spectrometry. Clin Chem 63:1008–1021

4. Carlier J, Diao X, Huestis MA (2018) Synthetic cannabinoid BB-22 (QUCHIC): human hepatocytes metabolism with liquid chromatography-high resolution mass spectrometry detection. J Pharm Biomed Anal 157:27–35

5. Carlier J, Diao X, Giorgetti R et al (2021) Pyrrolidinyl synthetic cathinones α-PHP and 4F-α-PVP metabolite profiling using human hepatocyte incubations. Int J Mol Sci 22:1–17

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