Optical Resolution ofdl-threo-2-(2,4-Difluorophenyl)-2-[1-(methylthio)ethyl]oxirane: Its Application to the Synthesis of SM-9164, a Biologically Active Enantiomer of Antifungal Agent SM-8668-Reference-Cited by-同舟云学术

Optical Resolution ofdl-threo-2-(2,4-Difluorophenyl)-2-[1-(methylthio)ethyl]oxirane: Its Application to the Synthesis of SM-9164, a Biologically Active Enantiomer of Antifungal Agent SM-8668

Published:1995-12 Issue:12 Volume:68 Page:3591-3598
ISSN:0009-2673
Container-title:Bulletin of the Chemical Society of Japan
language:en
Short-container-title:BCSJ

Author:

Miyauchi Hiroshi,Ohashi Naohito

Publisher

The Chemical Society of Japan

Subject

General Chemistry

Link

https://www.jstage.jst.go.jp/article/bcsj/68/12/68_12_3591/_pdf

Reference20 articles.

1. Stereoselective Synthesis of Antifungal Agentthreo-2-(2,4-Difluorophenyl)-3-methylsulfonyl-1-(1H-1,2,4-triazol-1-yl)-2-butanol (SM-8668)

2. Optically Active Antifungal Azoles. I. Synthesis and Antifungal Activity of (2R,3R)-2-(2,4-Difluorophenyl)-3-mercapto-1-(1H-1,2,4-triazol-1-yl)-2-butanol and Its Stereoisomers.

3. Triazole Antifungals. III. Stereocontrolled Synthesis of an Optically Active Triazolylmethyloxirane Precursor to Antifungal Oxazolidine Derivatives.

4. Synthesis and oral anti-fungal activity of novel 1,3-bis-(azolyl)-2-arylpropan-2-ols

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