Ibrutinib selectively and irreversibly targets EGFR (L858R, Del19) mutant but is moderately resistant to EGFR (T790M) mutant NSCLC Cells

Author:

Wu Hong12,Wang Aoli12,Zhang Wei3,Wang Beilei1,Chen Cheng1,Wang Wenchao1,Hu Chen1,Ye Zi4,Zhao Zheng1,Wang Li1,Li Xixiang1,Yu Kailin1,Liu Juan1,Wu Jiaxin12,Yan Xiao-E5,Zhao Peng5,Wang Jinhua6,Wang Chu4,Weisberg Ellen L.7,Gray Nathanael S.6,Yun Cai-Hong5,Liu Jing1,Chen Liang3,Liu Qingsong128

Affiliation:

1. High Magnetic Field Laboratory, Chinese Academy of Sciences, Hefei 230031, Anhui, P. R. China

2. University of Science and Technology of China, Hefei 230036, Anhui, P. R. China

3. Collaborative Innovation Center of Cancer Medicine, National Institute of Biological Sciences, Beijing, Beijing 102206, P.R. China

4. Synthetic and Functional Biomolecules Center, Beijing National Laboratory for Molecular Sciences, Key Laboratory of Bioorganic Chemistry and Molecular Engineering of Ministry of Education, College of Chemistry and Molecular Engineering, Peking-Tsinghua Center for Life Sciences, Peking University, Beijing 100871, P.R. China

5. Institute of Systems Biomedicine, Department of Biophysics, Beijing Key Laboratory of Tumor Systems Biology and Center for Molecular and Translational Medicine, School of Basic Medical Sciences, Peking University Health Science Center, Beijing 100191, P.R. China

6. Department of Cancer Biology, Dana-Farber Cancer Institute, and Department of Biological Chemistry & Molecular Pharmacology, Harvard Medical School, Boston, MA 02115, USA

7. Department of Medical Oncology, Dana Farber Cancer Institute, Harvard Medical School, Boston, MA 02115, USA

8. Hefei Science Center, Chinese Academy of Sciences, Hefei 230031, Anhui, P. R. China

Publisher

Impact Journals, LLC

Subject

Oncology

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