Chemical regulation of Kv7 channels: Diverse scaffolds, sites, and mechanisms of action-Reference-Cited by-同舟云学术

Chemical regulation of Kv7 channels: Diverse scaffolds, sites, and mechanisms of action

Published:2020-06-02 Issue:8 Volume:152 Page:
ISSN:0022-1295
Container-title:Journal of General Physiology
language:en
Short-container-title:

Author:

Kurata Harley T.¹^ORCID

Affiliation:

1. Department of Pharmacology, Alberta Diabetes Institute, University of Alberta, Edmonton, AB, Canada

Abstract

Kv7 channels are powerfully regulated by a wide variety of physiological and pharmacological signals. Larsson et al. describe the direct modulation of Kv7 channels by endocannabinoids and explore how combinations of Kv7 activators with distinct subtype specificities might lead to effective and selective drug cocktails.

Publisher

Rockefeller University Press

Subject

Physiology

Link

http://rupress.org/jgp/article-pdf/doi/10.1085/jgp.202012598/1044853/jgp_202012598.pdf

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