Synthesis of novel series of 3,5-disubstituted imidazo[1,2-<i>d</i>] [1,2,4]thiadiazoles involving S<sub>N</sub>Ar and Suzuki–Miyaura cross-coupling reactions-Reference-Cited by-同舟云学术

Synthesis of novel series of 3,5-disubstituted imidazo[1,2-d] [1,2,4]thiadiazoles involving S_NAr and Suzuki–Miyaura cross-coupling reactions

Published:2022 Issue:10 Volume:12 Page:6303-6313
ISSN:2046-2069
Container-title:RSC Advances
language:en
Short-container-title:RSC Adv.

Author:

Pescheteau Clémentine¹,Place Matthieu¹,Sava Alexandru¹²,Nunes Lea¹,Profire Lenuta³,Routier Sylvain¹^ORCID,Buron Frédéric¹^ORCID

Affiliation:

1. Institut de Chimie Organique et Analytique, ICOA, UMR CNRS 7311, Université d’Orléans, Orléans, France

2. Department of Analytical Chemistry, Faculty of Pharmacy, “Grigore T. Popa” University of Medicine and Pharmacy of Iasi, 16 University Street, 700115 Iasi, Romania

3. Department of Pharmaceutical Chemistry, Faculty of Pharmacy, “Grigore T. Popa” University of Medicine and Pharmacy of Iasi, 16 University Street, 700115 Iasi, Romania

Abstract

A convenient design of 3,5-disubstituted imidazo[1,2-d][1,2,4]thiadiazoles is reported from 2-mercaptoimidazole, which afforded a versatile platform that was then used to access a variety of original heterocycles.

Funder

Société Française de Radiologie

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemical Engineering,General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2022/RA/D1RA07208K

Reference28 articles.

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