Diastereoselective synthesis of functionalized tetrahydropyridazines containing indole scaffolds via an inverse-electron-demand aza-Diels–Alder reaction-Reference-Cited by-同舟云学术

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Diastereoselective synthesis of functionalized tetrahydropyridazines containing indole scaffolds via an inverse-electron-demand aza-Diels–Alder reaction

Published:2021 Issue:16 Volume:8 Page:4392-4398
ISSN:2052-4129
Container-title:Organic Chemistry Frontiers
language:en
Short-container-title:Org. Chem. Front.

Author:

Chen Taotao¹²³⁴⁵,Che Chao¹²³⁴⁵,Guo Zhefei¹²³⁴⁵,Dong Xiu-Qin¹²³⁴⁵^ORCID,Wang Chun-Jiang¹²³⁴⁵^ORCID

Affiliation:

1. Engineering Research Centre of Organosilicon Compounds & Materials

2. Ministry of Education

3. College of Chemistry and Molecular Sciences

4. Wuhan University

5. Wuhan

Abstract

A base-promoted and catalyst-free unprecedented inverse-electron-demand aza-Diels–Alder reaction between the in situ generated azoalkenes and 3-vinylindoles has been developed to afford tetrahydropyridazines containing indole scaffolds.

Funder

National Natural Science Foundation of China

Natural Science Foundation of Hubei Province

Natural Science Foundation of Jiangsu Province

Project 211

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2021/QO/D1QO00623A

Reference75 articles.

1. Heterocyclic Compounds as Inflammation Inhibitors

2. Recent Advance in Heterocyclic Organozinc and Organomanganese Compounds; Direct Synthetic Routes and Application in Organic Synthesis

3. Recent Advances in the Research of Heterocyclic Compounds as Antitubercular Agents

4. Sarcosine-Based Glycine Transporter Type-1 (GlyT-1) Inhibitors Containing Pyridazine Moiety: A Further Search for Drugs with Potential to Influence Schizophrenia Negative Symptoms

5. Discovery of Imidazo[1,2-b]pyridazine Derivatives: Selective and Orally Available Mps1 (TTK) Kinase Inhibitors Exhibiting Remarkable Antiproliferative Activity

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