On-resin synthesis of Lanreotide epimers and studies of their structure–activity relationships-Reference-Cited by-同舟云学术

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On-resin synthesis of Lanreotide epimers and studies of their structure–activity relationships

Published:2024 Issue:8 Volume:15 Page:2766-2772
ISSN:2632-8682
Container-title:RSC Medicinal Chemistry
language:en
Short-container-title:RSC Med. Chem.

Author:

Chowdhury Arnab¹^ORCID,Tripathi Nitesh Mani¹^ORCID,Jadav Rohit²,Gour Vinod¹,Purohit Parva²,Bandyopadhyay Anupam¹^ORCID

Affiliation:

1. Biomimetic Peptide Engineering Laboratory, Department of Chemistry, Indian Institute of Technology Ropar, Rupnagar, Punjab-140001, India

2. Kashiv BioSciences Pvt Ltd., Block-B, Sardar Patel Ring Rd, opp. Applewoods Township, Ahmedabad, Gujarat-382210, India

Abstract

This report demonstrates the rapid and clean on-resin assembly of disulfide, which enabled impurity and biological profiling of eight possible epimers of a somatostatin analog, lanreotide.

Funder

Indian Institute of Technology Ropar

Publisher

Royal Society of Chemistry (RSC)

Link

http://pubs.rsc.org/en/content/articlepdf/2024/MD/D4MD00338A

Reference23 articles.

1. Somatostatin analogs: does pharmacology impact antitumor efficacy?

2. Somatostatin-Dopamine Chimeric Molecules in Neuroendocrine Neoplasms

3. Peptide Receptor Targeting in Cancer: The Somatostatin Paradigm

4. Somatuline Autogel 60 mg, solution for injection in a prefilled syringe - Summary of Product Characteristics (SmPC) - (emc), https://www.medicines.org.uk/emc/product/4808/smpc#gref , (accessed 2 May 2023)

5. Lanreotide Depot: An Antineoplastic Treatment of Carcinoid or Neuroendocrine Tumors

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