Rapid access to N-(indol-2-yl)amides and N-(indol-3-yl)amides as unexplored pharmacophores-Reference-Cited by-同舟云学术

Rapid access to N-(indol-2-yl)amides and N-(indol-3-yl)amides as unexplored pharmacophores

Published:2017 Issue:3 Volume:15 Page:576-580
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Reekie Tristan A.¹²³,Wilkinson Shane M.¹²³,Law Vivian¹²³,Hibbs David E.⁴²³^ORCID,Ong Jennifer A.⁴²³,Kassiou Michael¹²³^ORCID

Affiliation:

1. School of Chemistry

2. University of Sydney

3. Australia

4. Faculty of Pharmacy

Abstract

Preparation of N-(indol-2-yl)amides and N-(indol-3-yl)amides are scarce in the scientific literature due to unstable intermediates impeding current reported syntheses.

Funder

National Health and Medical Research Council

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2017/OB/C6OB02622B

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