Second generation of thiazolylmannosides, FimH antagonists for E. coli-induced Crohn's disease-Reference-Cited by-同舟云学术

Second generation of thiazolylmannosides, FimH antagonists for E. coli-induced Crohn's disease

Published:2016 Issue:16 Volume:14 Page:3913-3925
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Chalopin T.¹²³⁴⁵,Alvarez Dorta D.¹²³⁴⁵,Sivignon A.⁶⁷⁸⁹,Caudan M.¹²³⁴⁵,Dumych T. I.¹⁰¹¹¹²⁹,Bilyy R. O.¹³¹⁴¹⁵,Deniaud D.¹²³⁴⁵,Barnich N.⁶⁷⁸⁹,Bouckaert J.¹⁰¹¹¹²⁹,Gouin S. G.¹²³⁴⁵

Affiliation:

1. LUNAM Université

2. CEISAM

3. Chimie Et Interdisciplinarité

4. Synthèse

5. Analyse

6. Clermont Université

7. UMR 1071 Inserm/Université d'Auvergne

8. 63000 Clermont-Ferrand

9. France

10. Unité de Glycobiologie Structurale et Fonctionnelle (UGSF)

11. UMR 8576 du CNRS

12. F-59655 Villeneuve d'Ascq Cedex

13. Danylo Halytsky Lviv National Medical University

14. Lviv

15. Ukraine

Abstract

The chemical stability of potentE. colianti-adhesives was improved by substitution of the anomeric nitrogen by short linkers.

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2016/OB/C6OB00424E

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5. The Bacterial Lectin FimH, a Target for Drug Discovery – Carbohydrate Inhibitors of Type 1 Fimbriae‐Mediated Bacterial Adhesion

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