Synthesis of C3-functionalized indole derivatives <i>via</i> Brønsted acid-catalyzed regioselective arylation of 2-indolylmethanols with guaiazulene-Reference-Cited by-同舟云学术

Synthesis of C3-functionalized indole derivatives via Brønsted acid-catalyzed regioselective arylation of 2-indolylmethanols with guaiazulene

Published:2022 Issue:7 Volume:20 Page:1510-1517
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Liu Yang¹^ORCID,Cao Meng¹,Zhang Shangxi¹,Wang Zhenxi¹^ORCID,Dai Xin¹,Jiang Xinde¹,Dong Yucheng¹,Fu Jie¹

Affiliation:

1. College of Science, Nanchang Institute of Technology, Nanchang 330099, People's Republic of China

Abstract

An efficient approach to the synthesis of guaiazulenyl C3-functionalized indoles with excellent regioselectivities via the Brønsted acid catalyzed arylation of 2-indolylmethanols is developed.

Funder

National Natural Science Foundation of China

Natural Science Foundation of Jiangxi Province

Key Research and Development Program of Jiangxi Province

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2022/OB/D1OB02384E

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