The synthesis, biological evaluation and structure–activity relationship of 2-phenylaminomethylene-cyclohexane-1,3-diones as specific anti-tuberculosis agents-Reference-Cited by-同舟云学术

The synthesis, biological evaluation and structure–activity relationship of 2-phenylaminomethylene-cyclohexane-1,3-diones as specific anti-tuberculosis agents

Published:2017 Issue:11 Volume:8 Page:2133-2141
ISSN:2040-2503
Container-title:MedChemComm
language:en
Short-container-title:Med. Chem. Commun.

Author:

Rather Muzafar Ahmad¹²³⁴⁵,Lone Ali Mohd⁶³⁴⁵,Teli Bisma⁶³⁴⁵⁷,Bhat Zubair Shanib¹²³⁴⁵,Singh Paramjeet⁸³⁹¹⁰,Maqbool Mubashir¹²³⁴⁵,Shairgojray Bashir Ahmad⁶³⁴⁵,Dar Mohd Jamal⁷¹¹⁸³⁹,Amin Shajrul¹²¹³¹⁴,Yousuf Syed Khalid⁶³⁴⁵⁷,Bhat Bilal A.⁶³⁴⁵⁷,Ahmad Zahoor¹²³⁴⁵^ORCID

Affiliation:

1. Clinical Microbiology and PK/PD Division

2. Clinical Microbiology PK/PD/Laboratory

3. CSIR-Indian Institute of Integrative Medicine

4. Srinagar

5. India-190005

6. Medicinal Chemistry Division

7. Academy of Scientific & Innovative Research (AcSIR)

8. Cancer Pharmacology Division

9. Jammu

10. India-180001

11. India

12. Department of Biochemistry

13. University of Kashmir

14. India-190006

Abstract

Synthetic interventions on previously identified hits; structure39was identified as the best lead againstMycobacterium tuberculosisH37Rv and was evaluated further.

Publisher

Royal Society of Chemistry (RSC)

Subject

Pharmaceutical Science,Biochemistry,Drug Discovery,Molecular Medicine,Pharmacology,Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2017/MD/C7MD00350A

Reference20 articles.

1. WHO Global tuberculosis report, 2016 , http://reliefweb.int/sites/reliefweb.int/files/resources/gtbr2016_main_text.pdf

2. HIV and COPD: a conspiracy of risk factors

3. Tuberculosis drug discovery in the post‐post‐genomic era

4. Resistance to rifampicin: a review

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