α-Amino bicycloalkylation through organophotoredox catalysis-Reference-Cited by-同舟云学术

α-Amino bicycloalkylation through organophotoredox catalysis

Published:2024 Issue:28 Volume:15 Page:10918-10925
ISSN:2041-6520
Container-title:Chemical Science
language:en
Short-container-title:Chem. Sci.

Author:

Nugent Jeremy¹,López-Francés Adrián²^ORCID,Sterling Alistair J.¹,Tay Min Yi¹,Frank Nils¹,Mousseau James J.³,Duarte Fernanda¹^ORCID,Anderson Edward A.¹^ORCID

Affiliation:

1. Department of Chemistry, Chemistry Research Laboratory, University of Oxford, 12 Mansfield Road, Oxford, OX1 3TA, UK

2. Department of Organic Chemistry I, Faculty of Pharmacy and Lascaray Research Center, University of the Basque Country, UPV/EHU, Paseo de la Universidad 7, 01006, Vitoria-Gasteiz, Spain

3. Pfizer Worldwide Research and Development, Eastern Point Road, Groton, Connecticut 06340, USA

Abstract

The organophotocatalysed-generation of α-amino radicals enables the synthesis of α-amino bicyclo[n.1.1]alkanes (n = 1, 3) under mild conditions by addition to the interbridgehead C–C bonds of [n.1.1]propellanes.

Funder

Engineering and Physical Sciences Research Council

H2020 Marie Skłodowska-Curie Actions

Eusko Jaurlaritza

Publisher

Royal Society of Chemistry (RSC)

Link

http://pubs.rsc.org/en/content/articlepdf/2024/SC/D4SC01368A

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