A gold-complex initiated functionalization of biologically active polyphenols applied to a <sup>18</sup>F-labeled chemical probe-Reference-Cited by-同舟云学术

A gold-complex initiated functionalization of biologically active polyphenols applied to a ¹⁸F-labeled chemical probe

Published:2023 Issue:29 Volume:21 Page:5990-5996
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Liu Ziyun¹^ORCID,Fukagawa Yuki¹,Yamano Masaharu¹,Tago Tetsuro²,Iwai Kumiko¹,Hirano Keiichi³,Kumazoe Motofumi⁴,Tachibana Hirofumi⁴^ORCID,Toyohara Jun²,Tanaka Hiroshi¹^ORCID

Affiliation:

1. Department of Chemical Science and Engineering, Tokyo Institute of Technology, 12-12-1-H101 Ookayama, Meguro, Tokyo, 152-8552, Japan

2. Research Team for Neuroimaging, Tokyo Metropolitan Institute for Geriatrics and Gerontology, 35-2 Sakae-cho, Itabashi-ku, Tokyo 173-0015, Japan

3. NMP Business Support Co., Ltd, Hyogo 669-1339, Japan

4. Division of Applied Biological Chemistry, Department of Bioscience and Biotechnology, Faculty of Agriculture, Kyushu University, Fukuoka, 819-0395, Japan

Abstract

A gold-complex initiated electrophilic aromatic substitution with amidomethyl 2-alknylbenzoates shortens the process to 18F-labeled polyphenol EGCG.

Funder

Japan Science and Technology Corporation

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2023/OB/D3OB00856H

Reference31 articles.

1. 67-kDa Laminin Receptor-Mediated Cellular Sensing System of Green Tea Polyphenol EGCG and Functional Food Pairing

2. A receptor for green tea polyphenol EGCG

3. The impact of the 67kDa laminin receptor on both cell-surface binding and anti-allergic action of tea catechins

4. Solid-Phase Synthesis of a Combinatorial Methylated (±)-Epigallocatechin Gallate Library and the Growth-Inhibitory Effects of these Compounds on Melanoma B16 Cells

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