Directed C(sp3)–H arylation of tryptophan: transformation of the directing group into an activated amide
Author:
Affiliation:
1. Philipps-Universität Marburg
2. Fachbereich Chemie
3. 35032 Marburg
4. Germany
Abstract
The aminoquinoline-directed C–H activation was used to synthezise unnatural tryptophans for solid phase peptide synthesis for the first time.
Publisher
Royal Society of Chemistry (RSC)
Subject
General Chemistry
Link
http://pubs.rsc.org/en/content/articlepdf/2019/SC/C9SC03440D
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