Synthesis, antimicrobial activity and molecular simulation of thiourea derivatives containing 6-carboalkoxybenzo[<i>d</i>]thiazole and <scp>d</scp>-glucose moieties-Reference-Cited by-同舟云学术

Synthesis, antimicrobial activity and molecular simulation of thiourea derivatives containing 6-carboalkoxybenzo[d]thiazole and d-glucose moieties

Published:2023 Issue:48 Volume:47 Page:22360-22376
ISSN:1144-0546
Container-title:New Journal of Chemistry
language:en
Short-container-title:New J. Chem.

Author:

Dinh Thanh Nguyen¹^ORCID,Son Hai Do¹²,Thi Kim Giang Nguyen¹²,Ngoc Toan Vu¹³,Thi Kim Van Hoang¹⁴,Minh Tri Nguyen¹³,Ngoc Toan Duong¹⁵

Affiliation:

1. Faculty of Chemistry, VNU University of Science (Vietnam National University, Ha Noi), 19 Le Thanh Tong, Hoan Kiem, Ha Noi, Vietnam

2. Institute of Science and Technology, Ministry of Public Security of Vietnam, 47 Pham Van Dong, Cau Giay, Ha Noi, Vietnam

3. Institute of New Technology, Military Institute of Science and Technology, 17 Hoang Sam, Cau Giay, Ha Noi, Vietnam

4. Faculty of Chemical Technology, Viet Tri University of Industry, Tien Kien, Lam Thao, Phu Tho, Vietnam

5. Faculty of Chemistry, Thai Nguyen University of Education, 20 Luong Ngoc Quyen, Thai Nguyen, Vietnam

Abstract

Substituted benzo[d]thiazole sulfonyl thioureas were synthesized. They exhibited antimicrobial activity, with some inhibiting Staphylococcus aureus DNA gyrase, DNA Topo IV, and dihydrofolate reductase. IFD, MM-GBSA and MD were performed on 6d/2XCS of S. aureus.

Publisher

Royal Society of Chemistry (RSC)

Subject

Materials Chemistry,General Chemistry,Catalysis

Link

http://pubs.rsc.org/en/content/articlepdf/2023/NJ/D3NJ04443B

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