Thiosuccinimide enabled S–N bond formation to access <i>N</i>-sulfenylated sulfonamide derivatives with synthetic diversity-Reference-Cited by-同舟云学术

Thiosuccinimide enabled S–N bond formation to access N-sulfenylated sulfonamide derivatives with synthetic diversity

Published:2024 Issue:5 Volume:22 Page:990-997
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Wang Peifeng¹^ORCID,Li Shan¹,Wen Huiling¹,Lei Yin¹,Huang Shujuan¹,Wang Zixiu¹,Su Jialong¹,Guan Wenxiang¹,Lei Jian¹^ORCID

Affiliation:

1. Key Laboratory of Prevention and Treatment of Cardiovascular and Cerebrovascular Disease of the Ministry of Education, Key Laboratory of Biomaterials and Biofabrication in Tissue Engineering of Jiangxi Province, College of Pharmacy, Gannan Medical University, Ganzhou 341000, PR China

Abstract

A thiosuccinimide enabled S–N cross-coupling strategy has been established for the intermolecular N-sulfenylation of clinically approved sulfa drugs under additive-free conditions.

Funder

National Natural Science Foundation of China

National College Students Innovation and Entrepreneurship Training Program

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2024/OB/D3OB01848B

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