Recent developments of imidazo[1,2-<i>a</i>]pyridine analogues as antituberculosis agents-Reference-Cited by-同舟云学术

Recent developments of imidazo[1,2-a]pyridine analogues as antituberculosis agents

Published:2023 Issue:4 Volume:14 Page:644-657
ISSN:2632-8682
Container-title:RSC Medicinal Chemistry
language:en
Short-container-title:RSC Med. Chem.

Author:

Samanta Sauvik¹^ORCID,Kumar Sumit¹,Aratikatla Eswar K.¹,Ghorpade Sandeep R.¹^ORCID,Singh Vinayak¹²^ORCID

Affiliation:

1. Holistic Drug Discovery and Development (H3D) Centre, University of Cape Town, Rondebosch 7701, South Africa

2. South African Medical Research Council Drug Discovery and Development Research Unit, Institute of Infectious Disease and Molecular Medicine, University of Cape Town, Rondebosch 7701, South Africa

Abstract

Here, we critically review anti-TB compounds of the imidazo[1,2-a]pyridine class by discussing their development based on the structure–activity relationship, mode-of-action, and various scaffold hopping strategies over the last decade.

Funder

Bill and Melinda Gates Foundation

South African Medical Research Council

Department of Science and Innovation, South Africa

National Research Foundation

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Drug Discovery,Pharmaceutical Science,Pharmacology,Molecular Medicine,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2023/MD/D3MD00019B

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